Добірка наукової літератури з теми "Internalization inhibitors"
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Статті в журналах з теми "Internalization inhibitors"
DiCello, Jesse J., Pradeep Rajasekhar, Emily M. Eriksson, Ayame Saito, Arisbel B. Gondin, Nicholas A. Veldhuis, Meritxell Canals, Simona E. Carbone та Daniel P. Poole. "Clathrin and GRK2/3 inhibitors block δ-opioid receptor internalization in myenteric neurons and inhibit neuromuscular transmission in the mouse colon". American Journal of Physiology-Gastrointestinal and Liver Physiology 317, № 2 (1 серпня 2019): G79—G89. http://dx.doi.org/10.1152/ajpgi.00085.2019.
Повний текст джерелаBigby, M., P. Wang, J. F. Fierro, and M. S. Sy. "Phorbol myristate acetate-induced down-modulation of CD4 is dependent on calmodulin and intracellular calcium." Journal of Immunology 144, no. 8 (April 15, 1990): 3111–16. http://dx.doi.org/10.4049/jimmunol.144.8.3111.
Повний текст джерелаvan Kerkhof, P., and G. J. Strous. "The ubiquitin-proteasome pathway regulates lysosomal degradation of the growth hormone receptor and its ligand." Biochemical Society Transactions 29, no. 4 (August 1, 2001): 488–93. http://dx.doi.org/10.1042/bst0290488.
Повний текст джерелаLuton, F., M. Buferne, J. Davoust, A. M. Schmitt-Verhulst, and C. Boyer. "Evidence for protein tyrosine kinase involvement in ligand-induced TCR/CD3 internalization and surface redistribution." Journal of Immunology 153, no. 1 (July 1, 1994): 63–72. http://dx.doi.org/10.4049/jimmunol.153.1.63.
Повний текст джерелаChen, Yang, Shan Wang, Xinan Lu, Haoran Zhang, Yan Fu, and Yongzhang Luo. "Cholesterol sequestration by nystatin enhances the uptake and activity of endostatin in endothelium via regulating distinct endocytic pathways." Blood 117, no. 23 (June 9, 2011): 6392–403. http://dx.doi.org/10.1182/blood-2010-12-322867.
Повний текст джерелаLazari, Maria de Fatima M., Xuebo Liu, Kazuto Nakamura, Jeffrey L. Benovic, and Mario Ascoli. "Role of G Protein-Coupled Receptor Kinases on the Agonist-Induced Phosphorylation and Internalization of the Follitropin Receptor." Molecular Endocrinology 13, no. 6 (June 1, 1999): 866–78. http://dx.doi.org/10.1210/mend.13.6.0289.
Повний текст джерелаAlmeida, Raul A., John R. Dunlap, and Stephen P. Oliver. "Binding of Host Factors Influences Internalization and Intracellular Trafficking ofStreptococcus uberisin Bovine Mammary Epithelial Cells." Veterinary Medicine International 2010 (2010): 1–8. http://dx.doi.org/10.4061/2010/319192.
Повний текст джерелаVan Hamme, Evelien, Hannah L. Dewerchin, Els Cornelissen, Bruno Verhasselt, and Hans J. Nauwynck. "Clathrin- and caveolae-independent entry of feline infectious peritonitis virus in monocytes depends on dynamin." Journal of General Virology 89, no. 9 (September 1, 2008): 2147–56. http://dx.doi.org/10.1099/vir.0.2008/001602-0.
Повний текст джерелаGoretzki, L., and B. M. Mueller. "Receptor-mediated endocytosis of urokinase-type plasminogen activator is regulated by cAMP-dependent protein kinase." Journal of Cell Science 110, no. 12 (June 15, 1997): 1395–402. http://dx.doi.org/10.1242/jcs.110.12.1395.
Повний текст джерелаHuang, Dianshuai, Qingjie Fan, Zhiyi Liu, Shuqin Zhang, Wei Huang, Hongrui Li, Chongyang Liang, and Fei Sun. "An Epitope on EGFR Loading Catastrophic Internalization Serve as a Novel Oncotarget for Hepatocellular Carcinoma Therapy." Cancers 12, no. 2 (February 16, 2020): 456. http://dx.doi.org/10.3390/cancers12020456.
Повний текст джерелаДисертації з теми "Internalization inhibitors"
Qian, Yanrong. "Internalization of Extracellular ATP in Cancer Cells and Development of New Generations of Anticancer Glucose Transport Inhibitors." Ohio University / OhioLINK, 2014. http://rave.ohiolink.edu/etdc/view?acc_num=ohiou1416411921.
Повний текст джерелаAlvear-Perez, Rodrigo. "Voies de signalisation activées lors de la stimulation du récepteur de l'apéline, responsables de l'effet hypotenseur de l'apéline." Electronic Thesis or Diss., Sorbonne Paris Cité, 2019. http://www.theses.fr/2019USPCB021.
Повний текст джерелаApeline is a vasoactive neuropeptide which plays a crucial role in maintaining water balance and cardiovascular functions. Laboratory studies on the effects of Aperlin-17 (K17F) and the K16P apelin fragment, corresponding to K17F deletion from phenylalanine (Phe) at its C-terminal part have shown the presence of this Phe is necessary for apelin to induce internalization of the Apelin receptor. Also cause a decrease in blood pressure. Subsequently, in the CHO cells expressing stably the murine receptor of the Apelin that the internalization of the Apelin receptor induced by K17F resulted in the activation of a second signaling pathway which is independent of the Gi protein, but dependent on beta-arrestin. This corresponds to the MAP kinase pathway (Mitogen Activator Protein Kinase), which could be involved in the hypotensive effect of the Apelin. My work consisted of characterizing a physiological model such as the rat kidney juxtamedullary afferent arterioles (JMAA), to study if the signaling pathway mediated by beta-arrestin was involved in the vasodilatory effect of K17F. Knowing that AngII induces vasoconstriction by increasing intracellular calcium mobilization ([Ca2+]i), we have showed by measuring variations in arteriolar diameter and [Ca2+]i, that when the Gi signaling pathway is blocked by pertussis toxin (PTX), the vasorelaxant effect induced by K17F is not modify. This data suggests that the vasorelaxing effect of K17F on AngII pre-contracted JMAAs is Gi-independent protein. In the presence of PTX and various internalization inhibitors the vasorelaxant effect induced by K17F on AngII-pre-contracted JMAAs is completely blocked. In addition, no significant decrease in [Ca2+]i mobilization is observed in the presence of PTX and these inhibitors, when K17F is applied to the plateau phase of the AngII-induced calcium response. This is in line with our hypothesis, that the vasorelaxing effect of K17F is Gi-independent protein and beta-arrestin-dependent. ApelineR is a potential therapeutic target for the treatment of heart failure and water retention. Knowing that the half-life of the aperitif in the bloodstream is approximatly one minute. Another aspect of my thesis was to develop metabolically stable K17F analogues by two different strategies. First, we have substituted each of the residues of the aperitif with its D-series enantiomer or a synthetic amino acid. Secondly, we added a fluoroalkyl chain to the N-terminal end of K17F. These two strategies have enabled us to obtain several compounds, the most active of which are P92 and LIT01-196. These retain pharmacological properties identical to those of K17F and have a plasma half-life significantly higher compared to the endogenous peptide. These two analogues have been shown to be active in vivo with the ability to reduce blood pressure and reduce vasopressin secretion in the blood leading to an increase in aqueous diuresis
Paradis, Justine. "Rôles non-canoniques des arrestines dans la signalisation et l’endocytose des récepteurs couplés aux protéines G." Thèse, 2017. http://hdl.handle.net/1866/20229.
Повний текст джерелаЧастини книг з теми "Internalization inhibitors"
Jiang, Fei, Naiguo Xing, Taiyong Lv, Zhanliang Sun, and Yan Zhao. "Effects of Eluting Volumes to Isolation Efficiencies in Manual Synthesis of Ga-68 Labelled FAPI-04." In Springer Proceedings in Physics, 270–75. Singapore: Springer Nature Singapore, 2023. http://dx.doi.org/10.1007/978-981-99-1023-6_25.
Повний текст джерелаТези доповідей конференцій з теми "Internalization inhibitors"
Barrott, Jared J., Aaron P. Smith, Takuya Osada, Nimmi Ramanujam, Michael R. Zalutsky, Kim Lyerly, and Timothy A. J. Haystead. "Abstract C86: Tethered Hsp90 inhibitors carrying optical or radioiodinated probes reveal selective internalization of ectopic Hsp90 in malignant breast tumor cells." In Abstracts: AACR-NCI-EORTC International Conference: Molecular Targets and Cancer Therapeutics--Oct 19-23, 2013; Boston, MA. American Association for Cancer Research, 2013. http://dx.doi.org/10.1158/1535-7163.targ-13-c86.
Повний текст джерелаYalcin, Huseyin, Hissa Al-Thani, and Samar Shurbaji. "Development and In Vivo Testing of Smart Nanoparticles for Enhanced Anti-Cancer Activity and Reduced Cardiotoxicity Associated with Tyrosine Kinase Inhibitors." In Qatar University Annual Research Forum & Exhibition. Qatar University Press, 2021. http://dx.doi.org/10.29117/quarfe.2021.0088.
Повний текст джерелаHutchinson, TE, S. Kuchibhotla, J. Zhang, ER Block та JM Patel. "Peptide Mediated Caveolar PKC-α Phosphorylation Inhibits Its Internalization in Lung Endothelial Cells." У American Thoracic Society 2009 International Conference, May 15-20, 2009 • San Diego, California. American Thoracic Society, 2009. http://dx.doi.org/10.1164/ajrccm-conference.2009.179.1_meetingabstracts.a6123.
Повний текст джерелаAllen, Fred D., Clara F. Asnes, Alan Wells, Elliot L. Elson, and Douglas A. Lauffenburger. "Alternative Pathways of Epidermal Growth Factor Receptor Mediated Contractile Force in NR6 Fibroblasts." In ASME 1999 International Mechanical Engineering Congress and Exposition. American Society of Mechanical Engineers, 1999. http://dx.doi.org/10.1115/imece1999-0403.
Повний текст джерелаHettmann, Thore, Matthias Schneider, Selam Ogbagabriel, Jiansong Xie, Gloria Juan, Susanne Hartmann, Robert Radinsky, and Daniel J. Freeman. "Abstract LB-306: U3-1287 (AMG 888), a fully human anti-HER3 mAb, inhibits HER3 activation and induces HER3 internalization and degradation." In Proceedings: AACR 101st Annual Meeting 2010‐‐ Apr 17‐21, 2010; Washington, DC. American Association for Cancer Research, 2010. http://dx.doi.org/10.1158/1538-7445.am10-lb-306.
Повний текст джерелаde Agostini, A., J. Marcum, and R. Rosenberg. "THE BINDING OF ANTITHROMBIN TO CAPILLARY ENDOTHELIAL CELLS GROWN IN VITRO." In XIth International Congress on Thrombosis and Haemostasis. Schattauer GmbH, 1987. http://dx.doi.org/10.1055/s-0038-1643343.
Повний текст джерелаWortinger, Mark A., Wei Zeng, Wei Jennifer Yang, Victoria Peek, Lei Yan, Jirong Lu, Chi-Kin Chow, et al. "Abstract 695: LA480, a c-Met antibody with neutralization and internalization properties, inhibits HGF-dependent and HGF-independent c-Met pathway activation and tumor growth." In Proceedings: AACR 101st Annual Meeting 2010‐‐ Apr 17‐21, 2010; Washington, DC. American Association for Cancer Research, 2010. http://dx.doi.org/10.1158/1538-7445.am10-695.
Повний текст джерелаDupuy, E., P. S. Rohrlich, and G. Tobelem. "HEPARIN STIMULATES FIBROBLAST GROWTH INDUCED BY PDGF." In XIth International Congress on Thrombosis and Haemostasis. Schattauer GmbH, 1987. http://dx.doi.org/10.1055/s-0038-1643750.
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