Articoli di riviste sul tema "Inhibition covalente"
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Aljoundi, Aimen, Ahmed El Rashedy, Patrick Appiah-Kubi e Mahmoud E. S. Soliman. "Coupling of HSP72 α-Helix Subdomains by the Unexpected Irreversible Targeting of Lysine-56 over Cysteine-17; Coevolution of Covalent Bonding". Molecules 25, n. 18 (16 settembre 2020): 4239. http://dx.doi.org/10.3390/molecules25184239.
Liu, S. Q., e P. A. Knauf. "Lys-430, site of irreversible inhibition of band 3 Cl- flux by eosin-5-maleimide, is not at the transport site". American Journal of Physiology-Cell Physiology 264, n. 5 (1 maggio 1993): C1155—C1164. http://dx.doi.org/10.1152/ajpcell.1993.264.5.c1155.
Yang, Jianhong, Yong Li, Wei Yan, Weimin Li, Qiang Qiu, Haoyu Ye e Lijuan Chen. "Covalent modification of Cys-239 in β-tubulin by small molecules as a strategy to promote tubulin heterodimer degradation". Journal of Biological Chemistry 294, n. 20 (2 aprile 2019): 8161–70. http://dx.doi.org/10.1074/jbc.ra118.006325.
Maksimenko, A. V., e R. Sh Beabealashvili. "Theoretical Grounding and Formation of Experimental Approaches to Hyaluronidase Structure Consolidation due to Its Computational Interactions with Shortchain Glycosaminoglycan Ligands". Биоорганическая химия 49, n. 4 (1 luglio 2023): 369–83. http://dx.doi.org/10.31857/s0132342323020161.
Bhatia, Sumeena, Steven C. Almo, Stanley G. Nathenson e Richard J. Hodes. "Dynamic equilibrium of B7-1 dimers and monomers is important for regulation of TCR/CD28 – mediated T cell activation (33.28)". Journal of Immunology 182, n. 1_Supplement (1 aprile 2009): 33.28. http://dx.doi.org/10.4049/jimmunol.182.supp.33.28.
Kuznetsova, Anastasiya, Philipp Klein e Till Opatz. "Halogenated 2,1,3-benzoxadiazoles as Potential Fluorescent Warheads for Covalent Protease Inhibitors". Proceedings 9, n. 1 (14 novembre 2018): 54. http://dx.doi.org/10.3390/ecsoc-22-05670.
Hognon, Cécilia, Marco Marazzi e Cristina García-Iriepa. "Atomistic-Level Description of the Covalent Inhibition of SARS-CoV-2 Papain-like Protease". International Journal of Molecular Sciences 23, n. 10 (23 maggio 2022): 5855. http://dx.doi.org/10.3390/ijms23105855.
Bisconte, Angelina, Ronald Hill, Michael Bradshaw, Erik Verner, David Finkle, Ken Brameld, Jens Funk, David Goldstein e Phil Nunn. "Efficacy in collagen induced arthritis models with a selective, reversible covalent Bruton’s tyrosine kinase inhibitor PRN473 is driven by durable target occupancy rather than extended plasma exposure (THER5P.904)". Journal of Immunology 194, n. 1_Supplement (1 maggio 2015): 139.6. http://dx.doi.org/10.4049/jimmunol.194.supp.139.6.
Beck, Philipp, Christian Dubiella e Michael Groll. "Covalent and non-covalent reversible proteasome inhibition". Biological Chemistry 393, n. 10 (1 ottobre 2012): 1101–20. http://dx.doi.org/10.1515/hsz-2012-0212.
Piestrzeniewicz, Mariola K., Dorota Wilmańska, Janusz Szemraj, Kazimierz Studzian e Marek Gniazdowski. "Interactions of Novel Morpholine and Hexamethylene Derivatives of Anthracycline Antibiotics with DNA". Zeitschrift für Naturforschung C 59, n. 9-10 (1 ottobre 2004): 739–48. http://dx.doi.org/10.1515/znc-2004-9-1020.
Müller, Patrick, Mergim Meta, Jan Laurenz Meidner, Marvin Schwickert, Jessica Meyr, Kevin Schwickert, Christian Kersten et al. "Investigation of the Compatibility between Warheads and Peptidomimetic Sequences of Protease Inhibitors—A Comprehensive Reactivity and Selectivity Study". International Journal of Molecular Sciences 24, n. 8 (13 aprile 2023): 7226. http://dx.doi.org/10.3390/ijms24087226.
Gerling, Katharina, Sabrina Ölschläger, Meltem Avci-Adali, Bernd Neumann, Ernst Schweizer, Christian Schlensak, Hans-Peter Wendel e Sandra Stoppelkamp. "A Novel C1-Esterase Inhibitor Oxygenator Coating Prevents FXII Activation in Human Blood". Biomolecules 10, n. 7 (13 luglio 2020): 1042. http://dx.doi.org/10.3390/biom10071042.
Stellmacher, Lena, Tatyana Sandalova, Sarah Schneider, Gunter Schneider, Georg A. Sprenger e Anne K. Samland. "Novel mode of inhibition byD-tagatose 6-phosphate through a Heyns rearrangement in the active site of transaldolase B variants". Acta Crystallographica Section D Structural Biology 72, n. 4 (24 marzo 2016): 467–76. http://dx.doi.org/10.1107/s2059798316001170.
Betori, Rick C., Yue Liu, Rama K. Mishra, Scott B. Cohen, Stephen J. Kron e Karl A. Scheidt. "Targeted Covalent Inhibition of Telomerase". ACS Chemical Biology 15, n. 3 (4 febbraio 2020): 706–17. http://dx.doi.org/10.1021/acschembio.9b00945.
Ghosh, Avick Kumar, Indranil Samanta, Anushree Mondal e Wenshe Ray Liu. "Covalent Inhibition in Drug Discovery". ChemMedChem 14, n. 9 (26 marzo 2019): 889–906. http://dx.doi.org/10.1002/cmdc.201900107.
Rao, AK, e MA Kowalska. "ADP-induced platelet shape change and mobilization of cytoplasmic ionized calcium are mediated by distinct binding sites on platelets: 5'- p-fluorosulfonylbenzoyladenosine is a weak platelet agonist". Blood 70, n. 3 (1 settembre 1987): 751–56. http://dx.doi.org/10.1182/blood.v70.3.751.751.
Rao, AK, e MA Kowalska. "ADP-induced platelet shape change and mobilization of cytoplasmic ionized calcium are mediated by distinct binding sites on platelets: 5'- p-fluorosulfonylbenzoyladenosine is a weak platelet agonist". Blood 70, n. 3 (1 settembre 1987): 751–56. http://dx.doi.org/10.1182/blood.v70.3.751.bloodjournal703751.
Bjij, Imane, Fisayo A. Olotu, Clement Agoni, Emmanuel Adeniji, Shama Khan, Ahmed El Rashedy, Driss Cherqaoui e Mahmoud E. S. Soliman. "Covalent Inhibition in Drug Discovery: Filling the Void in Literature". Current Topics in Medicinal Chemistry 18, n. 13 (4 ottobre 2018): 1135–45. http://dx.doi.org/10.2174/1568026618666180731161438.
Strelow, John M. "A Perspective on the Kinetics of Covalent and Irreversible Inhibition". SLAS DISCOVERY: Advancing the Science of Drug Discovery 22, n. 1 (5 ottobre 2016): 3–20. http://dx.doi.org/10.1177/1087057116671509.
Kilbourn, R., e G. Lopez-Berestein. "Protease inhibitors block the macrophage-mediated inhibition of tumor cell mitochondrial respiration." Journal of Immunology 144, n. 3 (1 febbraio 1990): 1042–45. http://dx.doi.org/10.4049/jimmunol.144.3.1042.
Colman, RW, WR Figures, LM Scearce, AM Strimpler, FX Zhou e AK Rao. "Inhibition of collagen-induced platelet activation by 5'-p- fluorosulfonylbenzoyl adenosine: evidence for an adenosine diphosphate requirement and synergistic influence of prostaglandin endoperoxides". Blood 68, n. 2 (1 agosto 1986): 565–70. http://dx.doi.org/10.1182/blood.v68.2.565.565.
Colman, RW, WR Figures, LM Scearce, AM Strimpler, FX Zhou e AK Rao. "Inhibition of collagen-induced platelet activation by 5'-p- fluorosulfonylbenzoyl adenosine: evidence for an adenosine diphosphate requirement and synergistic influence of prostaglandin endoperoxides". Blood 68, n. 2 (1 agosto 1986): 565–70. http://dx.doi.org/10.1182/blood.v68.2.565.bloodjournal682565.
Tian, Yafeng, Mi Zhang, Panpan Heng, Hua Hou e Baoshan Wang. "Computational Investigations on Reaction Mechanisms of the Covalent Inhibitors Ponatinib and Analogs Targeting the Extracellular Signal-Regulated Kinases". International Journal of Molecular Sciences 24, n. 20 (16 ottobre 2023): 15223. http://dx.doi.org/10.3390/ijms242015223.
Zhou, X. Edward, Kelly Suino-Powell, Chad R. Schultz, Bilal Aleiwi, Joseph S. Brunzelle, Jared Lamp, Irving E. Vega, Edmund Ellsworth, André S. Bachmann e Karsten Melcher. "Structural basis of binding and inhibition of ornithine decarboxylase by 1-amino-oxy-3-aminopropane". Biochemical Journal 478, n. 23 (6 dicembre 2021): 4137–49. http://dx.doi.org/10.1042/bcj20210647.
Kinoshita, T., A. W. Dodds, S. K. A. Law e K. Inoue. "The low C5 convertase activity of the C4A6 allotype of human complement component C4". Biochemical Journal 261, n. 3 (1 agosto 1989): 743–48. http://dx.doi.org/10.1042/bj2610743.
Stevic, Ivan, Howard H. W. Chan, Ankush Chander, Leslie R. Berry e Anthony K. C. Chan. "Covalently linking heparin to antithrombin enhances prothrombinase inhibition on activated platelets". Thrombosis and Haemostasis 109, n. 06 (2013): 1016–24. http://dx.doi.org/10.1160/th12-10-0766.
Sim, E., A. W. Dodds e A. Goldin. "Inhibition of the covalent binding reaction of complement component C4 by penicillamine, an anti-rheumatic agent". Biochemical Journal 259, n. 2 (15 aprile 1989): 415–19. http://dx.doi.org/10.1042/bj2590415.
Lu, Jia-Hui, Zhen Li, Jia-Hui Chen, Shu-Liang Li, Jie-Hao He, Song Gu, Bo-Wen Liu, Li Chen e Yu-Zhong Wang. "Adaptable Phosphate Networks towards Robust, Reprocessable, Weldable, and Alertable-Yet-Extinguishable Epoxy Vitrimer". Research 2022 (6 ottobre 2022): 1–12. http://dx.doi.org/10.34133/2022/9846940.
Ruddraraju, Kasi Viswanatharaju, e Zhong-Yin Zhang. "Covalent inhibition of protein tyrosine phosphatases". Molecular BioSystems 13, n. 7 (2017): 1257–79. http://dx.doi.org/10.1039/c7mb00151g.
Zhao, Yuguang, Fredrik Svensson, David Steadman, Sarah Frew, Amy Monaghan, Magda Bictash, Tiago Moreira et al. "Structural Insights into Notum Covalent Inhibition". Journal of Medicinal Chemistry 64, n. 15 (22 luglio 2021): 11354–63. http://dx.doi.org/10.1021/acs.jmedchem.1c00701.
Westover, Kenneth D., Pasi A. Jänne e Nathanael S. Gray. "Progress on Covalent Inhibition of KRASG12C". Cancer Discovery 6, n. 3 (marzo 2016): 233–34. http://dx.doi.org/10.1158/2159-8290.cd-16-0092.
Jacobs, Amy. "Covalent Inhibition of HIV Membrane Fusion". Biophysical Journal 96, n. 3 (febbraio 2009): 359a. http://dx.doi.org/10.1016/j.bpj.2008.12.1814.
Huang, Huang, Christina A. Howard, Sergei Zari, Hyo Je Cho, Shirish Shukla, Hao Li, Juliano Ndoj et al. "Covalent inhibition of NSD1 histone methyltransferase". Nature Chemical Biology 16, n. 12 (31 agosto 2020): 1403–10. http://dx.doi.org/10.1038/s41589-020-0626-6.
Amara, Neri, Roi Mashiach, Dotan Amar, Pnina Krief, Stéphane A. H. Spieser, Matthew J. Bottomley, Amir Aharoni e Michael M. Meijler. "Covalent Inhibition of Bacterial Quorum Sensing". Journal of the American Chemical Society 131, n. 30 (5 agosto 2009): 10610–19. http://dx.doi.org/10.1021/ja903292v.
Kentner, Taryn A., Leslie R. Berry e Anthony K. C. Chan. "Inhibition of Factor Xa in Prothrombinase Is Enhanced by Covalent Linkage of Antithrombin to Heparin." Blood 104, n. 11 (16 novembre 2004): 1051. http://dx.doi.org/10.1182/blood.v104.11.1051.1051.
NAGUMO, Yoko, Hideaki KAKEYA, Mitsuru SHOJI, Yujiro HAYASHI, Naoshi DOHMAE e Hiroyuki OSADA. "Epolactaene binds human Hsp60 Cys442 resulting in the inhibition of chaperone activity". Biochemical Journal 387, n. 3 (26 aprile 2005): 835–40. http://dx.doi.org/10.1042/bj20041355.
Jebaraj, Billy Michael Chelliah, Annika Müller, Rashmi Priyadharshini Dheenadayalan, Sascha Endres, Philipp M. Roessner, Felix Seyfried, Claudia Walliser et al. "Evaluation of vecabrutinib as a model for noncovalent BTK/ITK inhibition for treatment of chronic lymphocytic leukemia". Blood 139, n. 6 (10 febbraio 2022): 859–75. http://dx.doi.org/10.1182/blood.2021011516.
Wágner, Gábor, Tamara A. M. Mocking, Albert J. Kooistra, Inna Slynko, Péter Ábrányi-Balogh, György M. Keserű, Maikel Wijtmans, Henry F. Vischer, Iwan J. P. de Esch e Rob Leurs. "Covalent Inhibition of the Histamine H3 Receptor". Molecules 24, n. 24 (11 dicembre 2019): 4541. http://dx.doi.org/10.3390/molecules24244541.
Thøgersen, I. B., G. Salvesen, F. H. Brucato, S. V. Pizzo e J. J. Enghild. "Purification and characterization of an α-macroglobulin proteinase inhibitor from the mollusc Octopus vulgaris". Biochemical Journal 285, n. 2 (15 luglio 1992): 521–27. http://dx.doi.org/10.1042/bj2850521.
Shatan, Anastasiia B., Vitalii Patsula, Hana Macková, Andrii Mahun, Renáta Lehotská, Elena Piecková e Daniel Horák. "Silver-Sulfamethazine-Conjugated β-Cyclodextrin/Dextran-Coated Magnetic Nanoparticles for Pathogen Inhibition". Nanomaterials 14, n. 4 (17 febbraio 2024): 371. http://dx.doi.org/10.3390/nano14040371.
Lee, Jesang, e Seung Bum Park. "Extended Applications of Small-Molecule Covalent Inhibitors toward Novel Therapeutic Targets". Pharmaceuticals 15, n. 12 (27 novembre 2022): 1478. http://dx.doi.org/10.3390/ph15121478.
Walderveen, Maria Christina Van, Leslie Roy Berry, Helen Mary Atkinson e Anthony Kam Chuen Chan. "Covalent antithrombin-heparin effect on thrombin-thrombomodulin and activated protein C reaction with factor V/Va". Thrombosis and Haemostasis 103, n. 05 (2010): 910–19. http://dx.doi.org/10.1160/th09-07-0473.
Allgardsson, Anders, Lotta Berg, Christine Akfur, Andreas Hörnberg, Franz Worek, Anna Linusson e Fredrik J. Ekström. "Structure of a prereaction complex between the nerve agent sarin, its biological target acetylcholinesterase, and the antidote HI-6". Proceedings of the National Academy of Sciences 113, n. 20 (2 maggio 2016): 5514–19. http://dx.doi.org/10.1073/pnas.1523362113.
Lee, Chang-Uk, e Tom N. Grossmann. "Reversible Covalent Inhibition of a Protein Target". Angewandte Chemie International Edition 51, n. 35 (13 luglio 2012): 8699–700. http://dx.doi.org/10.1002/anie.201203341.
Ahmed, Vanessa F., Nunzio Bottini e Amy M. Barrios. "Covalent Inhibition of the Lymphoid Tyrosine Phosphatase". ChemMedChem 9, n. 2 (8 gennaio 2014): 296–99. http://dx.doi.org/10.1002/cmdc.201300404.
Stevic, Ivan, Howard H. W. Chan, Ankush Chander, Leslie R. Berry e Anthony K. C. Chan. "Inhibition of Platelet-Prothrombianse by a Covalent Antithrombin-Heparin Complex." Blood 120, n. 21 (16 novembre 2012): 2212. http://dx.doi.org/10.1182/blood.v120.21.2212.2212.
Zhou, Yuxin, Ji Tao, Dingshuainan Jin, Shiping Zhang, Yan He e Longlong Niu. "The Inhibition Effect and Mechnism of a Thiadiazole Derivative on Q235 Carbon Steel in 1 M HCl Solution". Applied Sciences 13, n. 4 (6 febbraio 2023): 2103. http://dx.doi.org/10.3390/app13042103.
Buneeva, O. A., L. N. Aksenova e A. E. Medvedev. "A Simple Approach for Pilot Analysis of Time-dependent Enzyme Inhibition: Discrimination Between Mechanism-based Inactivation and Tight Binding Inhibitor Behavior". Biomedical Chemistry: Research and Methods 3, n. 1 (2020): e00115. http://dx.doi.org/10.18097/bmcrm00115.
Wang, Qian, Guofeng Chen, Jian He, Jiameng Li, Muya Xiong, Haixia Su, Minjun Li, Hangchen Hu e Yechun Xu. "Structure-Based Design of Potent Peptidomimetic Inhibitors Covalently Targeting SARS-CoV-2 Papain-like Protease". International Journal of Molecular Sciences 24, n. 10 (11 maggio 2023): 8633. http://dx.doi.org/10.3390/ijms24108633.
Abdeldayem, Ayah, Yasir S. Raouf, Stefan N. Constantinescu, Richard Moriggl e Patrick T. Gunning. "Advances in covalent kinase inhibitors". Chemical Society Reviews 49, n. 9 (2020): 2617–87. http://dx.doi.org/10.1039/c9cs00720b.