Journal articles on the topic 'Small inhibitory compounds'
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Alvarez-Gonzalez, Juan Antonio, Robert Maul, Rahul M. Kohli, and Patricia J. Gearhart. "Small molecule inhibitors of Activation-Induced Deaminase." Journal of Immunology 200, no. 1_Supplement (May 1, 2018): 48.18. http://dx.doi.org/10.4049/jimmunol.200.supp.48.18.
Yan, Hua, Tomoko Chiba Mizutani, Nobuhiko Nomura, Tadakazu Takakura, Yoshihiro Kitamura, Hideka Miura, Masako Nishizawa, Masashi Tatsumi, Naoki Yamamoto, and Wataru Sugiura. "A Novel Small Molecular Weight Compound with a Carbazole Structure That Demonstrates Potent Human Immunodeficiency Virus Type-1 Integrase Inhibitory Activity." Antiviral Chemistry and Chemotherapy 16, no. 6 (December 2005): 363–73. http://dx.doi.org/10.1177/095632020501600603.
Asai, Takashi, Tsutomu Takeuchi, Jeff Diffenderfer, and L. David Sibley. "Identification of Small-Molecule Inhibitors of Nucleoside Triphosphate Hydrolase in Toxoplasma gondii." Antimicrobial Agents and Chemotherapy 46, no. 8 (August 2002): 2393–99. http://dx.doi.org/10.1128/aac.46.8.2393-2399.2002.
Patkar, Chinmay G., Martha Larsen, Michael Owston, Janet L. Smith, and Richard J. Kuhn. "Identification of Inhibitors of Yellow Fever Virus Replication Using a Replicon-Based High-Throughput Assay." Antimicrobial Agents and Chemotherapy 53, no. 10 (August 3, 2009): 4103–14. http://dx.doi.org/10.1128/aac.00074-09.
Han, Chun, Jiahong Ren, Feng Su, Xiaoqin Hu, Mengyao Li, Zhijun Wang, and Lintao Wu. "Hybrids of Quinoline and Anilinopyrimidine: Novel EGFRT790M Inhibitors with Antiproliferative Activity against Non-Small Cell Lung Cancer Cell Lines." Anti-Cancer Agents in Medicinal Chemistry 20, no. 6 (June 14, 2020): 724–33. http://dx.doi.org/10.2174/1871520620666200302113206.
Abramić, Marija, and Dejan Agić. "Survey of Dipeptidyl Peptidase III Inhibitors: From Small Molecules of Microbial or Synthetic Origin to Aprotinin." Molecules 27, no. 9 (May 7, 2022): 3006. http://dx.doi.org/10.3390/molecules27093006.
Noueiry, Amine O., Paul D. Olivo, Urszula Slomczynska, Yi Zhou, Ben Buscher, Brian Geiss, Michael Engle, et al. "Identification of Novel Small-Molecule Inhibitors of West Nile Virus Infection." Journal of Virology 81, no. 21 (August 22, 2007): 11992–2004. http://dx.doi.org/10.1128/jvi.01358-07.
Lefas, Georgia, and George Chaconas. "High-Throughput Screening Identifies Three Inhibitor Classes of the Telomere Resolvase from the Lyme Disease Spirochete." Antimicrobial Agents and Chemotherapy 53, no. 10 (July 13, 2009): 4441–49. http://dx.doi.org/10.1128/aac.00529-09.
Ercan-Fang, Nacide, Miriam R. Taylor, Judith L. Treadway, Carolyn B. Levy, Paul E. Genereux, E. Michael Gibbs, Virginia L. Rath, Younggil Kwon, Mary C. Gannon, and Frank Q. Nuttall. "Endogenous effectors of human liver glycogen phosphorylase modulate effects of indole-site inhibitors." American Journal of Physiology-Endocrinology and Metabolism 289, no. 3 (September 2005): E366—E372. http://dx.doi.org/10.1152/ajpendo.00264.2004.
Yoo, Jihye, Darong Kim, Jiyoung Park, Young-Kook Kim, Hea-Young Park Choo, and Hyun Ae Woo. "Novel Small Molecule Inhibitors Targeting the IL-6/STAT3 Pathway or IL-1β." Molecules 27, no. 9 (April 22, 2022): 2696. http://dx.doi.org/10.3390/molecules27092696.
Ramesh, Priyanka, and Shanthi Veerappapillai. "Designing Novel Compounds for the Treatment and Management of RET-Positive Non-Small Cell Lung Cancer—Fragment Based Drug Design Strategy." Molecules 27, no. 5 (February 28, 2022): 1590. http://dx.doi.org/10.3390/molecules27051590.
Gong, Mengdie, Mingyan Tu, Hongxia Sun, Lu Li, Lili Zhu, Honglin Li, Zhenjiang Zhao, and Shiliang Li. "Design, Synthesis, and Structure–Activity Relationship Study of Potent MAPK11 Inhibitors." Molecules 27, no. 1 (December 29, 2021): 203. http://dx.doi.org/10.3390/molecules27010203.
Tian, Tao, Guo-Ying Chen, Hao Zhang, and Feng-Qing Yang. "Personal Glucose Meter for α-Glucosidase Inhibitor Screening Based on the Hydrolysis of Maltose." Molecules 26, no. 15 (July 30, 2021): 4638. http://dx.doi.org/10.3390/molecules26154638.
Flaumenhaft, Robert, Lynn VerPlank, James R. Dilks, Price S. Blair, Albert Mairuhu, Joseph Negri, Jason Burbank, et al. "A Chemical Genetic Analysis of Platelet Activation." Blood 114, no. 22 (November 20, 2009): 4009. http://dx.doi.org/10.1182/blood.v114.22.4009.4009.
Choi, Ryan, Mowei Zhou, Roger Shek, Jesse W. Wilson, Logan Tillery, Justin K. Craig, Indraneel A. Salukhe, et al. "High-throughput screening of the ReFRAME, Pandemic Box, and COVID Box drug repurposing libraries against SARS-CoV-2 nsp15 endoribonuclease to identify small-molecule inhibitors of viral activity." PLOS ONE 16, no. 4 (April 22, 2021): e0250019. http://dx.doi.org/10.1371/journal.pone.0250019.
Ruseva, Nina, Hristina Sbirkova-Dimitrova, Mariyana Atanasova, Ana Marković, Žaklina Šmelcerović, Andrija Šmelcerović, Adriana Bakalova, and Emiliya Cherneva. "Synthesis and DNase I Inhibitory Properties of New Squaramides." Molecules 28, no. 2 (January 5, 2023): 538. http://dx.doi.org/10.3390/molecules28020538.
Huang, Yuting, Zhaoxing Li, Yuan Ma, Qianqian Wu, Jianping Kong, Lijuan Zhao, Shunxiang Li, and Juan Li. "Screening for Active Compounds of Acorus calamus against SARS-CoV-2 Viral Protease and Mechanism Prediction." Pharmaceuticals 17, no. 3 (March 1, 2024): 325. http://dx.doi.org/10.3390/ph17030325.
Sato, Yoshiaki, Ikuo Kashiwakura, Masaru Yamaguchi, Hironori Yoshino, Takeshi Tanaka, Ken Ikeda, Zhengmao Ye, Hirotsugu Komatsu, Takao Matsuzaki, and Masato Hosoda. "Discovery of a Novel Small-molecule Interleukin-6 Inhibitor Through Virtual Screening Using Artificial Intelligence." Medicinal Chemistry 18, no. 6 (July 2022): 694–700. http://dx.doi.org/10.2174/1573406418666211116144243.
Paiboonrungruang, chorlada. "Abstract 6237: Small molecule screen identifies pyrimethamine as an inhibitor of NRF2-driven esophageal hyperplasia." Cancer Research 83, no. 7_Supplement (April 4, 2023): 6237. http://dx.doi.org/10.1158/1538-7445.am2023-6237.
Jiang, Suping, Sean T. Prigge, Lan Wei, Yu-e. Gao, Thomas H. Hudson, Lucia Gerena, John B. Dame, and Dennis E. Kyle. "New Class of Small Nonpeptidyl Compounds BlocksPlasmodium falciparum Development In Vitro by Inhibiting Plasmepsins." Antimicrobial Agents and Chemotherapy 45, no. 9 (September 1, 2001): 2577–84. http://dx.doi.org/10.1128/aac.45.9.2577-2584.2001.
Moi, Davide, Alessandro Deplano, Andrea Angeli, Gianfranco Balboni, Claudiu T. Supuran, and Valentina Onnis. "Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity." Molecules 27, no. 17 (August 23, 2022): 5370. http://dx.doi.org/10.3390/molecules27175370.
Al-Sanea, Mohammad M. "Synthesis and biological evaluation of small molecule modulators of CDK8/Cyclin C complex with phenylaminoquinoline scaffold." PeerJ 8 (March 13, 2020): e8649. http://dx.doi.org/10.7717/peerj.8649.
Gao, Yinghong, Stephen P. Davies, Martin Augustin, Anna Woodward, Umesh A. Patel, Robert Kovelman, and Kevin J. Harvey. "A broad activity screen in support of a chemogenomic map for kinase signalling research and drug discovery." Biochemical Journal 451, no. 2 (March 28, 2013): 313–28. http://dx.doi.org/10.1042/bj20121418.
Cruz-Migoni, Abimael, Peter Canning, Camilo E. Quevedo, Carole J. R. Bataille, Nicolas Bery, Ami Miller, Angela J. Russell, Simon E. V. Phillips, Stephen B. Carr, and Terence H. Rabbitts. "Structure-based development of new RAS-effector inhibitors from a combination of active and inactive RAS-binding compounds." Proceedings of the National Academy of Sciences 116, no. 7 (January 25, 2019): 2545–50. http://dx.doi.org/10.1073/pnas.1811360116.
Ramshini, Hassan, Reza Tayebee, Alessandra Bigi, Francesco Bemporad, Cristina Cecchi, and Fabrizio Chiti. "Identification of Novel 1,3,5-Triphenylbenzene Derivative Compounds as Inhibitors of Hen Lysozyme Amyloid Fibril Formation." International Journal of Molecular Sciences 20, no. 22 (November 7, 2019): 5558. http://dx.doi.org/10.3390/ijms20225558.
Minhas, Richa, and Yogita Bansal. "iNOS inhibitors: Benzimidazole-coumarin derivatives to combat inflammation." European Journal of Chemistry 13, no. 3 (September 30, 2022): 307–18. http://dx.doi.org/10.5155/eurjchem.13.3.307-318.2282.
Chattopadhyay, Shrikanta, Alison L. Stewart, Siddhartha Mukherjee, Cherrie Huang, Kimberly A. Hartwell, Peter G. Miller, Leigh Carmody, et al. "Niche-Based Screening Identifies Novel Small Molecules That Overcome Stromal Effects in Multiple Myeloma." Blood 120, no. 21 (November 16, 2012): 571. http://dx.doi.org/10.1182/blood.v120.21.571.571.
Adachi, Ryutaro, Tsuyoshi Ishii, Shinichi Matsumoto, Takuya Satou, Junichi Sakamoto, and Tomohiro Kawamoto. "Discovery of Human Intestinal MGAT Inhibitors Using High-Throughput Mass Spectrometry." SLAS DISCOVERY: Advancing the Science of Drug Discovery 22, no. 4 (October 8, 2016): 360–65. http://dx.doi.org/10.1177/1087057116673181.
Mavridis, Evangelos, Eleftherios Bermperoglou, Eleni Pontiki, and Dimitra Hadjipavlou-Litina. "5-(4H)-Oxazolones and Their Benzamides as Potential Bioactive Small Molecules." Molecules 25, no. 14 (July 11, 2020): 3173. http://dx.doi.org/10.3390/molecules25143173.
Trenholme, Katharine, Linda Marek, Sandra Duffy, Gabriele Pradel, Gillian Fisher, Finn K. Hansen, Tina S. Skinner-Adams, et al. "Lysine Acetylation in Sexual Stage Malaria Parasites Is a Target for Antimalarial Small Molecules." Antimicrobial Agents and Chemotherapy 58, no. 7 (April 14, 2014): 3666–78. http://dx.doi.org/10.1128/aac.02721-13.
Zhao, Hongchuan, Pu Sun, Wei Guo, Yi Wang, Ao Zhang, Linghua Meng, and Chunyong Ding. "Discovery of Indoleamine 2,3-Dioxygenase 1 (IDO-1) Inhibitors Based on Ortho-Naphthaquinone-Containing Natural Product." Molecules 24, no. 6 (March 18, 2019): 1059. http://dx.doi.org/10.3390/molecules24061059.
Furbish, Amelia B., Ahmed S. Alford, Pieter Burger, Yuri K. Peterson, Tracy Murray-Stewart, Robert A. Casero, and Patrick M. Woster. "Identification and Characterization of Novel Small-Molecule SMOX Inhibitors." Medical Sciences 10, no. 3 (August 30, 2022): 47. http://dx.doi.org/10.3390/medsci10030047.
VENÄLÄINEN, Jarkko I., Risto O. JUVONEN, J. Arturo GARCIA-HORSMAN, Erik A. A. WALLÉN, Johannes A. M. CHRISTIAANS, Elina M. JARHO, Jukka GYNTHER, and Pekka T. MÄNNISTÖ. "Slow-binding inhibitors of prolyl oligopeptidase with different functional groups at the P1 site." Biochemical Journal 382, no. 3 (September 7, 2004): 1003–8. http://dx.doi.org/10.1042/bj20040992.
Kollár, Levente, Martina Gobec, Matic Proj, Lara Smrdel, Damijan Knez, Tímea Imre, Ágnes Gömöry, et al. "Fragment-Sized and Bidentate (Immuno)Proteasome Inhibitors Derived from Cysteine and Threonine Targeting Warheads." Cells 10, no. 12 (December 6, 2021): 3431. http://dx.doi.org/10.3390/cells10123431.
Nordio, Giulia, Francesco Piazzola, Giorgio Cozza, Monica Rossetto, Manuela Cervelli, Anna Minarini, Filippo Basagni, et al. "From Monoamine Oxidase Inhibition to Antiproliferative Activity: New Biological Perspectives for Polyamine Analogs." Molecules 28, no. 17 (August 29, 2023): 6329. http://dx.doi.org/10.3390/molecules28176329.
Moon, Sungho, Seon Yeon Cho, Minhye Kim, Soojeong Beak, Jinhyuk Kim, Yongchan Kim, Sungil Park, et al. "Abstract B142: Discovery of novel and potent TEAD inhibitors, orally available small molecules with anti-tumor activity in hippo pathway- dysregulated cancers." Molecular Cancer Therapeutics 22, no. 12_Supplement (December 1, 2023): B142. http://dx.doi.org/10.1158/1535-7163.targ-23-b142.
Rusina, Polina, Erik Gandalipov, Yana Abdusheva, Maria Panova, Alexandra Burdenkova, Vasiliy Chaliy, Maria Brachs, et al. "Imidazole-4-N-acetamide Derivatives as a Novel Scaffold for Selective Targeting of Cyclin Dependent Kinases." Cancers 15, no. 15 (July 25, 2023): 3766. http://dx.doi.org/10.3390/cancers15153766.
Francini, Cinzia, Francesca Musumeci, Anna Fallacara, Lorenzo Botta, Alessio Molinari, Roberto Artusi, Laura Mennuni, Adriano Angelucci, and Silvia Schenone. "Optimization of Aminoimidazole Derivatives as Src Family Kinase Inhibitors." Molecules 23, no. 9 (September 17, 2018): 2369. http://dx.doi.org/10.3390/molecules23092369.
Kulkarni, Amol A., Ayyiliath M. Sajith, Changwen Zhang, Jiukuan Hao, and J. Phillip Bowen. "Small molecule prevents inflammation in microglia by targeting the NLRP3 inflammasome." Journal of Immunology 204, no. 1_Supplement (May 1, 2020): 160.15. http://dx.doi.org/10.4049/jimmunol.204.supp.160.15.
Rampogu, Shailima, Ayoung Baek, Chanin Park, Shraddha Parate, Saravanan Parameswaran, Yohan Park, Baji Shaik, Ju Hyun Kim, Seok Ju Park, and Keun Woo Lee. "Discovery of Small Molecules that Target Vascular Endothelial Growth Factor Receptor-2 Signalling Pathway Employing Molecular Modelling Studies." Cells 8, no. 3 (March 21, 2019): 269. http://dx.doi.org/10.3390/cells8030269.
Gising, Johan, Saman Honarnejad, Maaike Bras, Gemma L. Baillie, Stuart P. McElroy, Philip S. Jones, Angus Morrison, Julia Beveridge, Mathias Hallberg, and Mats Larhed. "The Discovery of New Inhibitors of Insulin-Regulated Aminopeptidase by a High-Throughput Screening of 400,000 Drug-like Compounds." International Journal of Molecular Sciences 25, no. 7 (April 6, 2024): 4084. http://dx.doi.org/10.3390/ijms25074084.
Curreli, Francesca, Shahad Ahmed, Sofia M. B. Victor, Aleksandra Drelich, Siva S. Panda, Andrea Altieri, Alexander V. Kurkin, Chien-Te K. Tseng, Christopher D. Hillyer, and Asim K. Debnath. "Discovery of Highly Potent Fusion Inhibitors with Potential Pan-Coronavirus Activity That Effectively Inhibit Major COVID-19 Variants of Concern (VOCs) in Pseudovirus-Based Assays." Viruses 14, no. 1 (December 31, 2021): 69. http://dx.doi.org/10.3390/v14010069.
Elsawi, Ahmed E., Mai I. Shahin, Hager A. Elbendary, Tarfah Al-Warhi, Fatma E. Hassan, and Wagdy M. Eldehna. "1,2,4-Triazole-Tethered Indolinones as New Cancer-Fighting Small Molecules Targeting VEGFR-2: Synthesis, Biological Evaluations and Molecular Docking." Pharmaceuticals 17, no. 1 (January 8, 2024): 81. http://dx.doi.org/10.3390/ph17010081.
Porubin, Diana. "Inhibition of in Vitro Nitrosation of Nornicotine." Chemistry Journal of Moldova 2, no. 1 (December 2007): 78–82. http://dx.doi.org/10.19261/cjm.2007.02(1).11.
Montanari, Floriane, Anna Cseke, Katrin Wlcek, and Gerhard F. Ecker. "Virtual Screening of DrugBank Reveals Two Drugs as New BCRP Inhibitors." SLAS DISCOVERY: Advancing the Science of Drug Discovery 22, no. 1 (July 11, 2016): 86–93. http://dx.doi.org/10.1177/1087057116657513.
Zhang, Hao, Feng-Qing Yang, and Jian-Li Gao. "A Simple and Portable Personal Glucose Meter Method Combined with Molecular Docking for Screening of Lipase Inhibitors." Evidence-Based Complementary and Alternative Medicine 2022 (September 22, 2022): 1–9. http://dx.doi.org/10.1155/2022/4430050.
Alkhashrom, Sewar, Jintawee Kicuntod, Sigrun Häge, Johannes Schweininger, Yves A. Muller, Peter Lischka, Manfred Marschall, and Jutta Eichler. "Exploring the Human Cytomegalovirus Core Nuclear Egress Complex as a Novel Antiviral Target: A New Type of Small Molecule Inhibitors." Viruses 13, no. 3 (March 12, 2021): 471. http://dx.doi.org/10.3390/v13030471.
Yang, Cheng-Wei, Yung-Ning Yang, Po-Huang Liang, Chi-Min Chen, Wei-Liang Chen, Hwan-You Chang, Yu-Sheng Chao, and Shiow-Ju Lee. "Novel Small-Molecule Inhibitors of Transmissible Gastroenteritis Virus." Antimicrobial Agents and Chemotherapy 51, no. 11 (August 20, 2007): 3924–31. http://dx.doi.org/10.1128/aac.00408-07.
Liargkova, Thalia, Nikolaos Eleftheriadis, Frank Dekker, Efstathia Voulgari, Constantinos Avgoustakis, Marina Sagnou, Barbara Mavroidi, Maria Pelecanou, and Dimitra Hadjipavlou-Litina. "Small Multitarget Molecules Incorporating the Enone Moiety." Molecules 24, no. 1 (January 7, 2019): 199. http://dx.doi.org/10.3390/molecules24010199.
Zhang, Yan, and Niefang Yu. "Design, Synthesis and Biological Evaluation: 5-amino-1H-pyrazole-1- carbonyl derivatives as FGFR Inhibitors." Letters in Drug Design & Discovery 17, no. 11 (October 23, 2020): 1330–41. http://dx.doi.org/10.2174/1570180817999200608140628.