Journal articles on the topic 'Benzolactum'
Create a spot-on reference in APA, MLA, Chicago, Harvard, and other styles
Consult the top 50 journal articles for your research on the topic 'Benzolactum.'
Next to every source in the list of references, there is an 'Add to bibliography' button. Press on it, and we will generate automatically the bibliographic reference to the chosen work in the citation style you need: APA, MLA, Harvard, Chicago, Vancouver, etc.
You can also download the full text of the academic publication as pdf and read online its abstract whenever available in the metadata.
Browse journal articles on a wide variety of disciplines and organise your bibliography correctly.
Lam, Hon-Wah, Ka-Yi Man, Wai-Wing Chan, Zhongyuan Zhou, and Wing-Yiu Yu. "Rhodium(iii)-catalyzed formal oxidative [4 + 1] cycloaddition of benzohydroxamic acids and α-diazoesters. A facile synthesis of functionalized benzolactams." Org. Biomol. Chem. 12, no. 24 (2014): 4112–16. http://dx.doi.org/10.1039/c4ob00512k.
Full textDeVita, R. J., and M. J. Wyvratt. "Benzolactam growth hormone secretagogues." Drugs of the Future 21, no. 3 (1996): 273. http://dx.doi.org/10.1358/dof.1996.021.03.353289.
Full textRyu, Ilhyong, Takahide Fukuyama, and Takanobu Bando. "Electron-Transfer-Induced Intramolecular Heck Carbonylation Reactions Leading to Benzolactones and Benzolactams." Synthesis 50, no. 15 (May 29, 2018): 3015–21. http://dx.doi.org/10.1055/s-0037-1609964.
Full textBouillon, J. P., C. Atès, C. Maliverney, Z. Janousek, and H. G. Viehe. "β-TRIFLUOROACETYLATION OF LACTAMS AND BENZOLACTAMS." Organic Preparations and Procedures International 26, no. 2 (April 1994): 249–55. http://dx.doi.org/10.1080/00304949409458029.
Full textKhantikaew, Itsara, Masato Takahashi, Takuya Kumamoto, Noriyuki Suzuki, and Tsutomu Ishikawa. "Synthesis of (−)-benzolactam-V8 by application of asymmetric aziridination." Tetrahedron 68, no. 3 (January 2012): 878–82. http://dx.doi.org/10.1016/j.tet.2011.11.033.
Full textBock, Mark G., Robert M. DiPardo, Daniel F. Veber, Raymond S. L. Chang, Victor J. Lotti, Stephen B. Freedman, and Roger M. Freidinger. "Benzolactams as non-peptide cholecystokinin receptor ligands." Bioorganic & Medicinal Chemistry Letters 3, no. 5 (May 1993): 871–74. http://dx.doi.org/10.1016/s0960-894x(00)80683-6.
Full textMa, Dawei, Guoqiang Wang, Shaomeng Wang, Alan P. Kozikowski, Nancy E. Lewin, and Peter M. Blumberg. "Synthesis and protein kinase C binding activity of benzolactam-V7." Bioorganic & Medicinal Chemistry Letters 9, no. 10 (May 1999): 1371–74. http://dx.doi.org/10.1016/s0960-894x(99)00207-3.
Full textMokrosz, Maria J., Sijka Charakchieva-Minol, and Piotr Kowalski. "Benzolactam Derivatives and Their Affinity for α1- and α2- Adrenoreceptors." Archiv der Pharmazie 334, no. 1 (January 2001): 25–26. http://dx.doi.org/10.1002/1521-4184(200101)334:1<25::aid-ardp25>3.0.co;2-8.
Full textDe Vita, Robert J., Alison J. Frontier, William R. Schoen, Matthew J. Wyvratt, Michael H. Fisher, Kang Cheng, Wanda W. S. Chan, Bridget S. Butler, and Roy G. Smith. "Design and Synthesis of Potent Macrocyclic Benzolactam Growth Hormone Secretagogues." Helvetica Chimica Acta 80, no. 4 (June 30, 1997): 1244–59. http://dx.doi.org/10.1002/hlca.19970800421.
Full textBouillon, Jean-Philippe, Célâl Ates, Zdenek Janousek, and Heinz G. Viehe. "Trifluoromethylated heterocycles from β-trifluoroacetyl-lactams and -benzolactams." Tetrahedron Letters 34, no. 32 (August 1993): 5075–78. http://dx.doi.org/10.1016/s0040-4039(00)60679-2.
Full textBOUILLON, J. P., C. ATES, C. MALIVERNEY, Z. JANOUSEK, and H. G. VIEHE. "ChemInform Abstract: β-Trifluoroacetylation of Lactams and Benzolactams." ChemInform 25, no. 34 (August 19, 2010): no. http://dx.doi.org/10.1002/chin.199434096.
Full textIbarreta, Dolores, Miriam Duchén, Dawei Ma, Lixin Qiao, Alan P. Kozikowski, and René Etcheberrigaray. "Benzolactam (BL) enhances sAPP secretion in fibroblasts and in PC12 cells." NeuroReport 10, no. 5 (April 1999): 1035–40. http://dx.doi.org/10.1097/00001756-199904060-00026.
Full textRajapaksa, Naomi S., Alberto Gobbi, Joy Drobnick, Steven Do, Aleksandr Kolesnikov, Jun Liang, Yongsheng Chen, et al. "Discovery of Potent Benzolactam IRAK4 Inhibitors with Robust in Vivo Activity." ACS Medicinal Chemistry Letters 11, no. 3 (November 11, 2019): 327–33. http://dx.doi.org/10.1021/acsmedchemlett.9b00380.
Full textBOUILLON, J. P., C. ATES, Z. JANOUSEK, and H. G. VIEHE. "ChemInform Abstract: Trifluoromethylated Heterocycles from β-Trifluoroacetyllactams and -benzolactams." ChemInform 24, no. 47 (August 20, 2010): no. http://dx.doi.org/10.1002/chin.199347188.
Full textOrtega, Raquel, Harald Hübner, Peter Gmeiner, and Christian F. Masaguer. "Aromatic ring functionalization of benzolactam derivatives: New potent dopamine D3 receptor ligands." Bioorganic & Medicinal Chemistry Letters 21, no. 9 (May 2011): 2670–74. http://dx.doi.org/10.1016/j.bmcl.2010.12.083.
Full textMa, Dawei, Guoqiang Wang, Shaomeng Wang, Alan P. Kozikowski, Nancy E. Lewin, and Peter M. Blumberg. "ChemInform Abstract: Synthesis and Protein Kinase C Binding Activity of Benzolactam-V7." ChemInform 30, no. 37 (June 13, 2010): no. http://dx.doi.org/10.1002/chin.199937172.
Full textKozikowski, Alan P., Shaomeng Wang, Dawei Ma, Jiangchao Yao, Shakeel Ahmad, Robert I. Glazer, Krisztina Bogi, et al. "Modeling, Chemistry, and Biology of the Benzolactam Analogues of Indolactam V (ILV). 2. Identification of the Binding Site of the Benzolactams in the CRD2 Activator-Binding Domain of PKCδ and Discovery of an ILV Analogue of Improved Isozyme Selectivity." Journal of Medicinal Chemistry 40, no. 9 (April 1997): 1316–26. http://dx.doi.org/10.1021/jm960875h.
Full textTabata, Hidetsugu, Naoya Wada, Yuko Takada, Tetsuta Oshitari, Hideyo Takahashi, and Hideaki Natsugari. "Isolation and Characterization of Atropisomers of Seven-Membered-Ring Benzolactams." Journal of Organic Chemistry 76, no. 12 (June 17, 2011): 5123–31. http://dx.doi.org/10.1021/jo2008725.
Full textDing, Guangni, Xiaoyu Wu, Lili Jiang, Zhaoguo Zhang, and Xiaomin Xie. "Reduction of Benzolactams to Isoindoles via an Alkoxide-Catalyzed Hydrosilylation." Organic Letters 19, no. 22 (October 27, 2017): 6048–51. http://dx.doi.org/10.1021/acs.orglett.7b02739.
Full textEndo, Yasuyuki, Michihiro Ohno, Masaaki Hirano, Mayuko Takeda, Akiko Itai, and Koichi Shudo. "Chiral requirements for tumor promoters: Conformations and activity of benzolactams." Bioorganic & Medicinal Chemistry Letters 4, no. 3 (February 1994): 491–94. http://dx.doi.org/10.1016/0960-894x(94)80023-5.
Full textParsons, W. H., A. A. Patchett, M. K. Holloway, G. M. Smith, J. L. Davidson, V. J. Lotti, and R. S. L. Chang. "Cholecystokinin antagonists. Synthesis and biological evaluation of 3-substituted benzolactams." Journal of Medicinal Chemistry 32, no. 8 (August 1989): 1681–85. http://dx.doi.org/10.1021/jm00128a004.
Full textMa, Dawei, Tao Zhang, Guoqiang Wang, Alan P. Kozikowski, Nancy E. Lewin, and Peter M. Blumberg. "Synthesis of 7,8-disubstituted benzolactam-V8 and its binding to protein kinase C." Bioorganic & Medicinal Chemistry Letters 11, no. 2 (January 2001): 99–101. http://dx.doi.org/10.1016/s0960-894x(00)00609-0.
Full textDeVita, Robert J., William R. Schoen, Dong Ok, Louis Barash, Jeanette E. Brown, Michael H. Fisher, Paul Hodges, et al. "Benzolactam growth hormone secretagogues: replacements for the 2′-tetrazole moiety of L-692,429." Bioorganic & Medicinal Chemistry Letters 4, no. 15 (August 1994): 1807–12. http://dx.doi.org/10.1016/s0960-894x(01)80375-9.
Full textSasa, Hirotaka, Koyo Mori, Kotaro Kikushima, Yasuyuki Kita, and Toshifumi Dohi. "μ-Oxo-Hypervalent-Iodine-Catalyzed Oxidative C–H Amination for Synthesis of Benzolactam Derivatives." Chemical and Pharmaceutical Bulletin 70, no. 2 (February 1, 2022): 106–10. http://dx.doi.org/10.1248/cpb.c21-00980.
Full textMa, Dawei, Guozhi Tang, and Alan P. Kozikowski. "Synthesis of 7-Substituted Benzolactam-V8s and Their Selectivity for Protein Kinase C Isozymes." Organic Letters 4, no. 14 (July 2002): 2377–80. http://dx.doi.org/10.1021/ol026125l.
Full textNakagawa, Yu, Kazuhiro Irie, Akiko Masuda, and Hajime Ohigashi. "Synthesis, conformation and PKC isozyme surrogate binding of new lactone analogues of benzolactam-V8s." Tetrahedron 58, no. 11 (March 2002): 2101–15. http://dx.doi.org/10.1016/s0040-4020(02)00099-6.
Full textMa, Dawei, and Wenjun Tang. "Stereospecific synthesis of 9-substituted benzolactam-V8 from L-tyrosine via regioselective aromatic nitration." Tetrahedron Letters 39, no. 40 (October 1998): 7369–72. http://dx.doi.org/10.1016/s0040-4039(98)01598-6.
Full textOk, Hyun O., John L. Szumiloski, George A. Doldouras, William R. Schoen, Kang Cheng, Wanda W. S. Chan, Bridget S. Butler, Roy G. Smith, Michael H. Fisher, and Matthew J. Wyvratt. "Benzolactam growth hormone secretagogues: Replacement of the C-3 amide bond in L-692,429." Bioorganic & Medicinal Chemistry Letters 6, no. 24 (December 1996): 3051–56. http://dx.doi.org/10.1016/s0960-894x(96)00566-5.
Full textOrtega, Raquel, Enrique Raviña, Christian F. Masaguer, Filipe Areias, José Brea, María I. Loza, Laura López, Jana Selent, Manuel Pastor, and Ferran Sanz. "Synthesis, binding affinity and SAR of new benzolactam derivatives as dopamine D3 receptor ligands." Bioorganic & Medicinal Chemistry Letters 19, no. 6 (March 2009): 1773–78. http://dx.doi.org/10.1016/j.bmcl.2009.01.067.
Full textOrito, Kazuhiko, Akiyoshi Horibata, Takatoshi Nakamura, Harumi Ushito, Hideo Nagasaki, Motoki Yuguchi, Satoshi Yamashita, and Masao Tokuda. "Preparation of Benzolactams by Pd(OAc)2-Catalyzed Direct Aromatic Carbonylation." Journal of the American Chemical Society 126, no. 44 (November 2004): 14342–43. http://dx.doi.org/10.1021/ja045342+.
Full textDeVita, Robert J., William R. Schoen, Michael H. Fisher, Alison J. Frontier, Judith M. Pisano, Matthew J. Wyvratt, Kang Cheng, et al. "Benzolactam growth hormone secretagogues: Carboxamides as replacements for the 2′-tetrazole moiety of L-692,429." Bioorganic & Medicinal Chemistry Letters 4, no. 18 (September 1994): 2249–54. http://dx.doi.org/10.1016/s0960-894x(00)80080-3.
Full textDeVita, Robert J., William R. Schoen, George A. Doldouras, Michael H. Fisher, Matthew J. Wyvratt, Kang Cheng, Wanda W. S. Chan, Bridget S. Butler, and Roy G. Smith. "Heterocyclic analogs of the benzolactam nucleus of the non-peptidic growth hormone secretagogue L-692,429." Bioorganic & Medicinal Chemistry Letters 5, no. 12 (June 1995): 1281–86. http://dx.doi.org/10.1016/0960-894x(95)00209-c.
Full textMa, Dawei, Tao Zhang, Guoqiang Wang, Alan P. Kozikowski, Nancy E. Lewin, and Peter M. Blumberg. "ChemInform Abstract: Synthesis of 7,8-Disubstituted Benzolactam-V8 and Its Binding to Protein Kinase C." ChemInform 32, no. 17 (April 24, 2001): no. http://dx.doi.org/10.1002/chin.200117166.
Full textGuo, Xiao-Yan, Run-Peng Qi, De-Gang Xu, Xu-Hua Liu, and Xiao Yang. "Structural and energetic insight into the interactions between the benzolactam inhibitors and tumor marker HSP90α." Computational Biology and Chemistry 58 (October 2015): 182–91. http://dx.doi.org/10.1016/j.compbiolchem.2015.07.013.
Full textLópez, Blanca, Aleix Rodriguez, David Santos, Joan Albert, Xavier Ariza, Jordi Garcia, and Jaume Granell. "Preparation of benzolactams by Pd(ii)-catalyzed carbonylation of N-unprotected arylethylamines." Chem. Commun. 47, no. 3 (2011): 1054–56. http://dx.doi.org/10.1039/c0cc03478a.
Full textOrito, Kazuhiko, Mamoru Miyazawa, Ryo Kanbayashi, Takashi Tatsuzawa, Masao Tokuda, and Hiroshi Suginome. "Benzolactams. 4. Reaction of 3‘,4‘- or 4‘,5‘-Dialkoxy-Substituted 1-(2‘-Bromobenzyl)-2-ethoxycarbonyl-1,2,3,4-tetrahydroisoquinolines with Alkyllithium. 1,2 and 1,4 Additions of Alkyllithium to Benzolactams." Journal of Organic Chemistry 65, no. 22 (November 2000): 7495–500. http://dx.doi.org/10.1021/jo000749s.
Full textEndo, Yasuyuki, Shunji Takehana, Michihiro Ohno, Paul E. Driedger, Silvia Stabel, Miho Y. Mizutani, Nobuo Tomioka, Akiko Itai, and Koichi Shudo. "Clarification of the Binding Mode of Teleocidin and Benzolactams to the Cys2 Domain of Protein Kinase Cδ by Synthesis of Hydrophobically Modified, Teleocidin-Mimicking Benzolactams and Computational Docking Simulation." Journal of Medicinal Chemistry 41, no. 9 (April 1998): 1476–96. http://dx.doi.org/10.1021/jm970704s.
Full textKamochi, Yasuko, and Yasuo Watanabe. "Studies on the Synthesis of Benzolactam Rings. II. Synthesis of 1,4-Dihydro-3(2H)-iaoquinolinone Derivatives." HETEROCYCLES 26, no. 9 (1987): 2385. http://dx.doi.org/10.3987/r-1987-09-2385.
Full textOhwada, Tomohiko, Hiroaki Kurouchi, and Yuko Otani. "Facile Synthesis of 5- to 7-Membered Benzolactam Compounds via Strongly Facilitated Electrophilic Aromtic Substitution Reaction†." HETEROCYCLES 93, no. 2 (2016): 705. http://dx.doi.org/10.3987/com-15-s(t)60.
Full textOKABE, Sachiko, Naoko SUEOKA, Atsumasa KOMORI, Masami SUGANUMA, Yasuyuki ENDO, Koichi SHUDO, and Hirota FUJIKI. "Twist Form of Teleocidin Derivatives is Active in in vivo Tumor Promotion by (-)-Benzolactam-V8-310." Biological & Pharmaceutical Bulletin 21, no. 5 (1998): 465–68. http://dx.doi.org/10.1248/bpb.21.465.
Full textMa, Dawei, Wenjun Tang, Alan P. Kozikowski, Nancy E. Lewin, and Peter M. Blumberg. "General and Stereospecific Route to 9-Substituted, 8,9-Disubstituted, and 9,10-Disubstituted Analogues of Benzolactam-V8." Journal of Organic Chemistry 64, no. 17 (August 1999): 6366–73. http://dx.doi.org/10.1021/jo990605h.
Full textDuffey, Matthew O., Tricia J. Vos, Ruth Adams, Jennifer Alley, Justin Anthony, Cynthia Barrett, Indu Bharathan, et al. "Discovery of a Potent and Orally Bioavailable Benzolactam-Derived Inhibitor of Polo-Like Kinase 1 (MLN0905)." Journal of Medicinal Chemistry 55, no. 1 (December 5, 2011): 197–208. http://dx.doi.org/10.1021/jm2011172.
Full textOK, H. O., J. L. SZUMILOSKI, G. A. DOLDOURAS, W. R. SCHOEN, K. CHENG, W. W. S. CHAN, B. S. BUTLER, R. G. SMITH, M. H. FISHER, and M. J. WYVRATT. "ChemInform Abstract: Benzolactam Growth Hormone Secretagogues: Replacement of the C-3 Amide Bond in L-692,429." ChemInform 28, no. 24 (August 3, 2010): no. http://dx.doi.org/10.1002/chin.199724172.
Full textMa, Dawei, Guozhi Tang, and Alan P. Kozikowski. "ChemInform Abstract: Synthesis of 7-Substituted Benzolactam-V8s and Their Selectivity for Protein Kinase C Isozymes." ChemInform 33, no. 48 (May 18, 2010): no. http://dx.doi.org/10.1002/chin.200248171.
Full textMA, D., and W. TANG. "ChemInform Abstract: Stereospecific Synthesis of 9-Substituted Benzolactam-V8 from L-Tyrosine via Regioselective Aromatic Nitration." ChemInform 29, no. 51 (June 18, 2010): no. http://dx.doi.org/10.1002/chin.199851261.
Full textFu, Ying, Ruijuan Li, Mingpeng Li, Yongyan Zhang, Yuxia Zhang, and Tianyu Yang. "Photocatalyzed Dehydroxylative Amination of Phenols: A Ring-Expansion Approach for Medium-Sized Benzolactams." Organic Letters 23, no. 21 (October 11, 2021): 8317–21. http://dx.doi.org/10.1021/acs.orglett.1c03053.
Full textPrado, Maria A. F., Ricardo J. Alves, José D. Souza Filho, Rosemeire B. Alves, Maria T. C. Pedrosa, Renata F. Prado, and André A. G. Faraco. "Synthesis of benzolactams by 11-endo selective aryl radical cyclisation of 2-iodobenzamides." Journal of the Chemical Society, Perkin Transactions 1, no. 12 (2000): 1853–57. http://dx.doi.org/10.1039/b002416n.
Full textOrito, Kazuhiko, Mamoru Miyazawa, Ryo Kanbayashi, Takashi Tatsuzawa, Masao Tokuda, and Hiroshi Suginome. "ChemInform Abstract: Benzolactams. Part 4. Reaction of 3′,4′- or 4′,5′-Dialkoxy-Substituted 1-(2′-Bromobenzyl)-2-ethoxycarbonyl-1,2,3,4-tetrahydroisoquinolines with Alkyllithium. 1,2 and 1,4 Additions of Alkyllithium to Benzolactams." ChemInform 32, no. 12 (March 20, 2001): no. http://dx.doi.org/10.1002/chin.200112151.
Full textNakagawa, Yu, Kazuhiro Irie, Ryo C. Yanagita, Hajime Ohigashi, Ken-ichiro Tsuda, Kaori Kashiwagi, and Naoaki Saito. "Design and Synthesis of 8-Octyl-benzolactam-V9, a Selective Activator for Protein Kinase Cε and η." Journal of Medicinal Chemistry 49, no. 9 (May 2006): 2681–88. http://dx.doi.org/10.1021/jm050857c.
Full textHUANG, Li-Li, Da-Wei MA, and Zong-Xiang XIA. "Molecular Modeling of Interactions of the Benzolactam-V8 Modulators with the Cys2 Domain of Protein Kinase Cδ." Chinese Journal of Chemistry 25, no. 10 (October 2007): 1434–38. http://dx.doi.org/10.1002/cjoc.200790265.
Full text